普立肽Plitidepsin(Aplidin)
称号 | 普立肽Aplidin(Plitidepsin) |
---|---|
CAS No. | 137219-37-5 |
规格 | mg/g/kg |
纯度 | ≥98% |
储存 | -20°C |
份子量 | 1110.357 |
序列布局 | (2S)-N-[(2R)-1-[[(3S,6S,8S,12S,13R,16S,17R,20S,23S)-13-[(2S)-butan-2-yl]-12-hydroxy-20-[(4-methoxyphenyl)methyl]-6,17,21-trimethyl-3-(2-methylpropyl)-2,5,7,10,15,19,22-heptaoxo-8-propan-2-yl-9,18-dioxa-1,4,14,21-tetrazabicyclo[21.3.0]hexacosan-16-yl]amino |
产物简述 |
Plitidepsin(又称)是从红色念珠菌海鞘中提取的一种化合物。今朝正在停止临床实验测试。它是被称为去甲肾上腺素具备抗肿瘤、抗病毒和免疫按捺活性。它在减少胰腺癌、胃癌、膀胱癌和前线腺癌的肿瘤方面显现出杰出的远景。 Plitidepsin (also known as dehydrodidemnin B) is a chemical compound extracted from the ascidian Aplidium albicans. It is currently undergoing clinical trial testing. It is a member of the class of compounds known as didemnins.plitidepsin exhibits antitumor, antiviral and immunosuppressive activities. It shows promise in shrinking tumors in pancreatic, stomach, bladder, and prostate cancers. |